Selpercatinib - LOXO-292

Based on 6 reference(s) in Google Scholar 8 10 6

Axon 3195

CAS [2361241-23-6]

MF C29H31N7O3
MW 525.60

  • Purity: 99%
  • Soluble in 0.1N HCl(aq) and DMSO

Selpercatinib

Description

Selpercatinib is a potent, highly selective, ATP-competitive RET inhibitor with an IC50 value of 4 nM (KIF5B-RET). Selpercatinib demonstrated potent and selective anti-RET activity preclinically against human cancer cell lines harboring endogenous RET gene alterations.

KEYWORDS: Selpercatinib | supplier | RET inhibitor | LOXO-292 | LOXO292 | LOXO 292 | CAS [2361241-23-6] | GDNF | RET | Inhibitor | Receptors

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10 mg €130.00 In Stock
50 mg €450.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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