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AZD1656

Based on 13 reference(s) in Google Scholar 8 10 13

Axon 3062

CAS [919783-22-5]

MF C24H26N6O5
MW 478.50

Purity: 99%
Optical purity: Optically pure
Soluble in DMSO

AZD1656

Description

AZD1656 is a potent, selective glucokinase (GK) activator that progressed to Phase IIb trials for the treatment of type 2 diabetes.

KEYWORDS: AZD1656 | supplier | GK activator | AZD-1656 | AZD 1656 | CAS [919783-22-5] | Glucose | Glucokinase | Activator | Enzymes | Type 2 Diabetes

MJ Waring et al. Property based optimisation of glucokinase activators - discovery of the phase IIb clinical candidate AZD1656. Med. Chem. Commun., 2012, 3, 1077-1081.

D McKerrecher et al. Design and development of the glucokinase activator AZD1656. ACS Symposium Series (2018), 1307(Complete Accounts of Integrated Drug Discovery and Development: Recent Examples from the Pharmaceutical Industry, Volume 1), 185-220.

Cell Signaling & Oncology Diabetes & Metabolism Glucokinase EC 2.7.1.2

Glucokinase (GK) activator

Chemical name

(S)-3-(5-(Azetidine-1-carbonyl)pyrazin-2-yloxy)-5-(1-methoxypropan-2-yloxy)-N-(5-methylpyrazin-2-yl)benzamide

Parent CAS No.

[919783-22-5]

Order

Size	Unit Price	Stock
5 mg	€165.00	In Stock
25 mg	€660.00	In Stock

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