BAY-598

Based on 2 reference(s) in Google Scholar 8 10 2

Axon 2635

CAS [1906919-67-2]

MF C22H20Cl2F2N6O3
MW 525.34

  • Purity: 98%
  • Optical purity: 99% e.e.
  • Soluble in DMSO

BAY-598

Description

BAY-598 is a potent, selective, and cell-active, substrate-competitive inhibitor of SMYD2 (IC50 values of 27 nM and 58 nM for biochemical and cellular activity, respectively). BAY-598 also shows PAR1 antagonism, but there is a greater than 50-fold selectivity for SMYD2 relative to PAR1.

KEYWORDS: BAY-598 | supplier | SMYD2 inhibitor | BAY598 | BAY 598 | CAS [1906919-67-2] | Histone | HMTase | Inhibitor | Enzymes | SET | MYND | Protein Methylation | Chemical Probe | Apoptosis | Protein Lysine Methyltransferase | SET and MYND Domain Containing Protein 2

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Size Unit Price Stock
2 mg €110.00 In Stock
5 mg €160.00 In Stock
25 mg €560.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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