Brexpiprazole dihydrochloride - OPC 34712 dihydrochloride

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 2335

CAS [2512192-75-3]

MF C25H27N3O2S.2HCl
MW 506.49

  • Purity: 98%
  • Soluble in DMSO

Brexpiprazole dihydrochloride


Drug candidate in clinical development for psychiatric disorders with high affinity for h5-HT1A (partial agonist), h5-HT2A (antagonist), hD2L (partial agonist), hα1B (antagonist) and hα2C-adrenergic (antagonist) receptors (Ki values <1 nM). Brexpiprazole also shows substantial affinity (Ki <5 nM) for hD3, h5-HT2B, h5-HT7, hα1A and hα1D adrenergic receptors, and moderate affinity for hH1 (Ki =19 nM).
Size Unit Price Stock
5 mg €135.00 In Stock
25 mg €475.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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