EMPA

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 2012

CAS [680590-49-2]

MF C23H26N4O4S
MW 454.54

Purity: 99%
Soluble in DMSO and Ethanol

EMPA

Description

Highly potent and selective orexin type 2 (OX2) receptor antagonist, with Ki values of >900 and 1 nM for OX1 and OX2 receptors respectively

P Malherbe et al. Biochemical and behavioural characterization of EMPA, a novel high-affinity, selective antagonist for the OX2 receptor. Br. J. Pharmacol. 2009, 156, 1326–1341.

TE Scammell and CJ Winrow. Orexin Receptors: Pharmacology and Therapeutic Opportunities. Annu. Rev. Pharmacol. Toxicol. 2011. 51:243–66.

Orexin type 2 (OX2) receptor antagonist

Chemical name

N-ethyl-2-(N-(6-methoxypyridin-3-yl)-2-methylphenylsulfonamido)-N-(pyridin-3-ylmethyl)acetamide

Parent CAS No.

[680590-49-2]

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EMPA

Description

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