GMC 2-118
Axon 1084
CAS:
256227-78-8
Purity:
98%
- No solubility data
- MF: C29H31N5O5S
- MW: 561.65
Description
Selective 5-HT1B antagonist, very potent in function assays
More Information
| Parent CAS No. | 256227-78-8 |
|---|---|
| Chemical Name | Methanesulfonic acid 4-{[2'-methyl-4'-(5-methyl-[1,3,4]oxadiazol-2-yl)-biphenyl-4-carbonyl]-amino}-2-(4-methyl-piperazin-1-yl)-phenyl ester |
| SMILES | N1(C2=CC(=CC=C2OS(C)(=O)=O)NC(=O)C2C=CC(=CC=2)C2C(C)=CC(C3OC(C)=NN=3)=CC=2)CCN(C)CC1 |
| MFCD | MFCD10565906 |
| InChi | InChI=1S/C29H31N5O5S/c1-19-17-23(29-32-31-20(2)38-29)9-11-25(19)21-5-7-22(8-6-21)28(35)30-24-10-12-27(39-40(4,36)37)26(18-24)34-15-13-33(3)14-16-34/h5-12,17-18H,13-16H2,1-4H3,(H,30,35) |
| InChiKey | FRSKIBLQHPOBGH-UHFFFAOYSA-N |
| CID | 10530932 |
| Short Description | 5-HT1B antagonist |
References
- Y Liao et al. New selective and potent 5-HT1B/1D or 5-HT1B antagonists: chemistry and pharmacological evaluation of GR127935-like compounds. J. Med. Chem. 2000, 43, 517-525.
- JW Clitherow et al. Evolution of a novel series of [(N,N-dimethylamino)propyl]- and piperazinylbenzalides as the first selective 5-HT1D antagonists. J. Med. Chem. 1994, 37, 2253.
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