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HTH-01-015

Axon 4391
CAS:  1613724-42-7
Purity:  99%
  • Soluble in 0.1N HCl(aq), DMSO and EtOH
  • MF:  C26H28N8O
  • MW:  468.55

Description

HTH-01-015 is a selective inhibitor of NUAK1 (IC50 value of 100 nM) which inhibits NUAK1 with >100-fold higher potency than NUAK2.

More Information

Parent CAS No. 1613724-42-7
Chemical Name 2,9-Dimethyl-7-methyl-5-(1-(4-piperidyl)-4-pyrazolylamino)-2,4,6,9-tetraazatetracyclo[9.8.0.0³,⁸.0¹³,¹⁸]nonadeca-1(19),3,5,7,11,13(18),14,16-octaen-10-one
Short Description NUAK1 inhibitor

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