EPZ005687 hydrochloride
- EPZ015938 hydrochloride
Axon 4137
- Parent CAS: 1396772-26-1
Purity:
99%
- Soluble in DMSO
- MF: C32H37N5O3.HCl
- MW: 576.13
Description
EPZ005687 is a potent and selective small molecule inhibitor of histone methyltransferase EZH2 ( Ki = 24 nM). It has greater than 500-fold selectivity against 15 other protein methyltransferases and has 50-fold selectivity against the closely related enzyme EZH1.
More Information
| Parent CAS No. | 1396772-26-1 |
|---|---|
| Chemical Name | 1-Cyclopentyl-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-6-(4-(morpholinomethyl)phenyl)-1H-indazole-4-carboxamide hydrochloride |
| extra_info | Sold in collaboration with Chemietek |
| MFCD | N.A. |
| Short Description | EZH2 HMTase inhibitor |
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