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DYRK1A inhibitor compound 11

Name: DYRK1A inhibitor compound 11
SKU: 4056

Axon 4056

CAS: 2814486-79-6

Purity: 98%

Soluble in 0.1N HCl(aq), DMSO and EtOH

MF: C12H12N6
MW: 240.26

Description

DYRK1A inhibitor compound 11 is a highly selective and ligand-efficient DYRK1A inhibitor with an IC50 value of 220 nM.

More Information

Certificate of Analysis (B2)

Material Safety Data Sheet (B2)

Certificate of Analysis

Material Safety Data Sheet

DYRK

Parent CAS No.	2814486-79-6
Chemical Name	N,N-Dimethyl-4-(pyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-amine
MFCD	N.A.
Short Description	Dyrk1A inhibitor

DYRK1A inhibitor compound 11 Dyrk1A inhibitor CAS 2814486-79-6 Axon Medchem Axon 4056 Non Selective (Phosphorylation substrates) DYRK Inhibitor Enzymes Alzheimer’s disease Down's syndrome Diabetes Supplier Vendor

References

SH Henderson et al. Discovery and Characterization of Selective and Ligand-Efficient DYRK Inhibitors. J Med Chem. 2021 Aug 12;64(15):11709-11728.

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DYRK1A inhibitor compound 11

Description

More Information

Certificate of Analysis

Material Safety Data Sheet

References

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