RTK class I; EC 2.7.10.1

27 Item(s)

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Axon ID Name Description From price
3040 Abivertinib Potent oral, irreversible, third-generation EGFR TKI with selectivity for mutant EGFRs €95.00
1986 AST 1306 tosylate ErbB2 and EGFR inhibitor €90.00
4074 AZ5104 EGFR inhibitor Inquire
2563 AZD3759 Potent, orally active, brain-penetrant, EGFR tyrosine kinase inhibitor €85.00
2342 AZD9291 Potent oral, irreversible, third-generation EGFR TKI with selectivity for mutant EGFRs €95.00
1544 BIBW 2992 EGFR and ErbB-2/HER2 tyrosine kinase inhibitor €50.00
3853 BMS-599626 Potent and selective EGFR and ErbB2 inhibitor Inquire
1433 CI 1033 EGFR tyrosine kinase inhibitor €60.00
1537 CP 724714 ErbB-2/HER2 kinase inhibitor €80.00
3235 Dacomitinib Potent irreversible pan-HER inhibitor €60.00
2680 EAI045 Allosteric EGFR inhibitor (L858R/T790M-specific) €105.00
1760 EGFR Inhibitor [879127-07-8] Highly selective EGFR tyrosine kinase inhibitor €120.00
3192 EMI48 Inhibitor of EGFR triple mutants €120.00
1128 Erlotinib hydrochloride EGFR tyrosine kinase inhibitor €70.00
1393 Gefitinib EGFR tyrosine kinase inhibitor €70.00
1395 Lapatinib ditosylate EGFR and ErbB-2/HER2 tyrosine kinase inhibitor €80.00
1526 Neratinib EGFR and ErbB-2/HER2 tyrosine kinase inhibitor €80.00
2955 NSC 228155 EGFR tyrosine kinase activator; Inhibitor of KIX-KID interaction €75.00
4144 Olmutinib Orally bioavailable and irreversible Tyrosine Kinase Inhibitor Inquire
1632 OSI 420 EGFR tyrosine kinase inhibitor €90.00
1665 Pelitinib EGFR tyrosine kinase inhibitor €90.00
2920 Poziotinib Irreversible pan-HER inhibitor €95.00
2053 TAK 165 ErbB2/HER2 kinase inhibitor €60.00
3232 TAK-788 Potent and selective EGFR and ErbB-2/HER2 tyrosine kinase inhibitor €70.00
4272 TAS2940 Orally active, brain-penetrable, and irreversible pan-ERBB inhibitor €110.00
3802 TAS6417 EGFR inhibitor Inquire
1506 WZ 4002 EGFR kinase inhibitor (T790M specific) €70.00

27 Item(s)

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