GA-017

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 4102

CAS [2351906-74-4]

MF C18H21N3O4
MW 343.38

  • Purity: 98%
  • Soluble in DMSO and EtOH

GA-017

Description

GA-017 is the first potent LATS1/2 inhibitor that exhibits sufficient growth-promoting effect on a variety of cell types under 3D conditions. GA-017 inhibited the activity of large tumor suppressor kinase 1 and 2 (LATS1/2), components of the Hippo pathway that mediate phosphorylation of YAP/TAZ, with IC50 values of 4.10 nM and 3.92 nM for LATS1 and LATS2, respectively.

KEYWORDS: GA-017 | Supplier | LATS1/2 inhibitor | GA017 | GA 017 | CAS [2351906-74-4] | Non Selective (Serine peptide bonds) | Inhibitor | Enzymes | Transcription Factors

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Size Unit Price Stock
5 mg €140.00 In Stock
25 mg €490.00 In Stock
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Size Unit Price Stock
2 x 5 mg €240.00 In Stock
2 x 25 mg €780.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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