CaMKIIα inhibitor compound 4d

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 3700

CAS [3031484-08-6]

MF C14H11ClO4
MW 278.69

Purity: 98%
Soluble in 0.1N NaOH(aq), DMSO and EtOH

CaMKIIα inhibitor compound 4d

Description

CaMKIIα inhibitor compound 4d is a high-affinity ligand with enhanced pharmacokinetic properties interacting strongly with the CaMKII α hub domain (Ki value of 0.027 μM). Powerful tool for potential allosteric regulation of CaMKII α kinase activity.

Y Tian et al. Discovery and Optimization of 5-Hydroxy-Diclofenac toward a New Class of Ligands with Nanomolar Affinity for the CaMKIIα Hub Domain. J Med Chem. 2022 May 12;65(9):6656-6676.

CNS CaMK EC 2.7.11.17

Ca2+/calmodulin-dependent protein kinase II α (CaMKIIα) inhibitor

Chemical name

2-(2-(2-Chlorophenoxy)-5-hydroxyphenyl)acetic acid

Parent CAS No.

[3031484-08-6]

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CaMKIIα inhibitor compound 4d

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CaMKIIα inhibitor compound 4d

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