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Repaglinide
- AG-EE 623ZW
Axon 3365
CAS:
135062-02-1
- Optical Purity: Optically pure
- Soluble in 0.1N NaOH(aq) and DMSO
- MF: C27H36N2O4
- MW: 452.59
Description
Antidiabetic; KATP channel blocker. Repaglinide was found to bind with low affinity (Kd of 59 nM) to SUR1 alone, but with high affinity (increased approximately 150-fold) when SUR1 was co-expressed with Kir6.2 (Kd value of 0.42 nM).
More Information
| Parent CAS No. | 135062-02-1 |
|---|---|
| Chemical Name | (S)-2-Ethoxy-4-(2-(3-methyl-1-(2-(piperidin-1-yl)phenyl)butylamino)-2-oxoethyl)benzoic acid |
| SMILES | C1C=C([C@H](CC(C)C)NC(=O)CC2C=CC(C(=O)O)=C(OCC)C=2)C(N2CCCCC2)=CC=1 |&1:3,r| |
| MFCD | N.A. |
| InChi | InChI=1S/C27H36N2O4/c1-4-33-25-17-20(12-13-22(25)27(31)32)18-26(30)28-23(16-19(2)3)21-10-6-7-11-24(21)29-14-8-5-9-15-29/h6-7,10-13,17,19,23H,4-5,8-9,14-16,18H2,1-3H3,(H,28,30)(H,31,32)/t23-/m0/s1 |
| InChiKey | FAEKWTJYAYMJKF-QHCPKHFHSA-N |
| CID | 65981 |
| Short Description | KATP channel blocker |
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