BChE inhibitor 8012-9656

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 3297

CAS [446266-84-8]

MF C21H17N7O2
MW 399.41

  • Purity: 98%
  • Soluble in DMSO
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BChE inhibitor 8012-9656

Description

BChE inhibitor 8012-9656 is a highly potent, selective and brain-penetrant inhibitor of butyrylcholinsterase with IC50 values of 0.18 and 0.32 μM for eqBChE and hBChE, respectively. BChE in a noncompetitive manner and could occupy the binding pocket forming diverse interactions with the target.

KEYWORDS: BChE inhibitor 8012-9656 | Supplier | BChE inhibitor | 8012 9656 | CAS [446266-84-8] | Choline-based esters | BChE | Inhibitor | Enzymes | Alzheimer’s disease

Highly potent, selective and brain-penetrant BChE inhibitor

Chemical name

2-(2-(4-Amino-1,2,5-oxadiazol-3-yl)-1H-benzo[d]imidazol-1-yl)-N-(2-methylquinolin-6-yl)acetamide

Parent CAS No.

[446266-84-8]

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5 mg €140.00 In Stock
25 mg €490.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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