ML-792

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 3109

CAS [1644342-14-2]

MF C21H23BrN6O5S
MW 551.41

  • Purity: 99%
  • Optical purity: Optically pure
  • Soluble in 0.1N NaOH(aq), 0.1N HCl(aq) and DMSO
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ML-792

Description

ML-792 is a potent and selective SUMO-activating enzyme (SAE) inhibitor with IC50 values of 0.003 μM and 0.011 μM when SUMO1 or SUMO2 was used as the ubiquitin-like protein (UBL), respectively. ML-792 selectively blocks total SUMOylation, thus decreasing cancer cell proliferation.

KEYWORDS: ML-792 | supplier | SAE inhibitor | ML792 | ML 792 | CAS [1644342-14-2] | Non Selective (Ubiquitin peptides) | Ubiquitin Ligase (E1) | Inhibitor | Enzymes | SUMO

Potent and selective inhibitor of SUMO-activating enzyme (SAE)

Chemical name

((1R,2S,4R)-4-(5-(1-(3-Bromobenzyl)-1H-pyrazole-3-carbonyl)pyrimidin-4-ylamino)-2-hydroxycyclopentyl)methyl sulfamate

Parent CAS No.

[1644342-14-2]

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5 mg €145.00 In Stock
25 mg €475.00 In Stock
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Size Unit Price Stock
2 x 5 mg €240.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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