GSK626616

Based on 3 reference(s) in Google Scholar 8 10 3

Axon 2970

CAS [1025821-33-3]

MF C18H10Cl2N4OS
MW 401.27

  • Purity: 99%
  • Soluble in DMSO
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GSK626616

Description

GSK626616 is a potent, orally bioavailable inhibitor of DYRK3 with an IC50 value of 0.7 nM. GSK626616 inhibits other members of the DYRK family, e.g., DYRK1A and DYRK2, with similar potency and with an approximate 20-fold selectivity versus the next most potently inhibited kinase, casein kinase 2.

KEYWORDS: GSK626616 | Supplier | DYRK3 inhibitor | GSK 626616 | GSK-626616 | CAS [1025821-33-3] | [2734473-05-1] | [1092362-47-4] | Non Selective (Phosphorylation Substrates) | DYRK | Inhibitor | Enzymes

Potent, orally bioavailable inhibitor of DYRK3

Chemical name

(5Z)-2-(2,6-dichlorophenylimino)-5-(quinoxalin-6-ylmethylene)thiazolidin-4-one

Parent CAS No.

[1025821-33-3]

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5 mg €120.00 In Stock
25 mg €420.00 In Stock
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2 x 5 mg €180.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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