Y 29794 tosylate

Based on 3 reference(s) in Google Scholar 8 10 3

Axon 2911

CAS [143984-17-2]

MF C30H42N2O4S3
MW 590.86

  • Purity: 99%
  • Soluble in DMSO
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Y 29794 tosylate

Description

Y 29794 tosylate is an orally active, potent and specific prolyl endopeptidase (PPCE) inhibitor that is easily penetrable into the brain. Y-29794 tosylate selectively and competitively inhibited rat brain PPCE in a reversible manner with a Ki value of 0.95 nM. Moreover, Y 29794 tosylate exhibited potent inhibitory activity with an IC50 value of 3.0 nM for both brain crude extract and partially purified enzyme fraction.

KEYWORDS: Y 29794 tosylate | supplier | PPCE inhibitor | Y29794 tosylate | Y-29794 tosylate | CAS [143984-17-2] | [129184-48-1] | [146794-84-5] | Non Selective (Serine Peptide Bonds) | Prolyl endopeptidase | Inhibitor | Enzymes | Alzheimer's disease

Orally active, brain penetrant, potent and specific prolyl endopeptidase (PPCE) inhibitor

Chemical name

(2-(8-(Dimethylamino)octylthio)-6-isopropylpyridin-3-yl)(thiophen-2-yl)methanone tosylate

Parent CAS No.

[129184-48-1]

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10 mg €125.00 In Stock
50 mg €450.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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