Based on 1 reference(s) in Google Scholar 8 10 1

Axon 2889

CAS [885898-58-8]

MF C21H19N3
MW 313.40

  • Purity: 99%
  • Soluble in DMSO



VA012 is a positive allosteric modulator of the serotonin 5-HT2C receptor with an EC50 value of 16 nM. VA012 exhibits enhanced efficacy dose-dependently, no significant off-target activities, and low competition with the endogenous agonist or other orthosteric ligands.

KEYWORDS: VA012 | supplier | PAM of 5-HT2C | VA 012 | VA-012 | CAS [885898-58-8] | Serotonin | 5-HT2C | PAM | Receptors | Obesity

Size Unit Price Stock
10 mg €105.00 In Stock
50 mg €315.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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