SB 747651A - SB 747651 tetrahydrochloride

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Axon 1897

CAS [2108968-31-4]

MF C16H22N8O.4HCl
MW 488.24

  • Purity: 98%
  • Soluble in water and DMSO

SB 747651A

Description

Potent MSK inhibitor; In vitro, SB-747651A inhibits MSK1 with an IC50 value of 11 nM; In cells, SB-747651A fully inhibited MSK activity at 5-10 μM.SB-747651A exhibited improved selectivity over H89 and Ro 31-8220 and therefore represents a useful tool to study MSK function in cells
Inhibitor of MSK1

Chemical name

4-(1-ethyl-7-((piperidin-4-ylamino)methyl)-1H-imidazo[4,5-c]pyridin-2-yl)-1,2,5-oxadiazol-3-amine tetrahydrochloride

Parent CAS No.

[607372-46-3]

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5 mg €120.00 In Stock
25 mg €420.00 In Stock
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2 x 5 mg €180.00 In Stock
2 x 25 mg €700.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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