Tolvaptan - OPC 41061

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1591

CAS [150683-30-0]

MF C26H25ClN2O3
MW 448.94

Purity: 99%
Soluble in DMSO

Tolvaptan

Description

A highly potent, oral and selective antagonist of vasopressin V2 receptor

Y Yamamura et al. OPC-41061, a Highly Potent Human Vasopressin V2-Receptor Antagonist: Pharmacological Profile and Aquaretic Effect by Single and Multiple Oral Dosing in Rats. J. Pharmacol. Exp. Ther. 1998, 287(3), 860-867.

T Hirano et al. Effects of the V2-Receptor Antagonist OPC-41061 and the Loop Diuretic Furosemide Alone and in Combination in Rats. JPET 2000, 292(1), 288-294.

RW Schrier et al. Tolvaptan, a Selective Oral Vasopressin V2-Receptor Antagonist, for Hyponatremia. N Engl J Med 2006, 355, 2099-2112.

Cardiovascular CNS A6 Vasopressin (V)

Vasopressin (V2) antagonist

Chemical name

N-(4-(7-chloro-5-hydroxy-2,3,4,5-tetrahydro-1H-benzo[b]azepine-1-carbonyl)-3-methylphenyl)-2-methylbenzamide

Parent CAS No.

[150683-30-0]

Order

Size	Unit Price	Stock
10 mg	€110.00	In Stock
50 mg	€330.00	In Stock

Need more? Bulk Inquiry

Related Products

Axon ID	Name	Description
1114	SSR 149415	Vasopressin (V1B) antagonist	€130.00
1256	SR 49059	Vasopressin (V1A) antagonist	€130.00
2146	Fedovapagon	Selective vasopressin V2 receptor agonist	€140.00
1867	Vasopressin antagonist 1867	Orally available and selective V1b receptor antagonist	€150.00

Customer Support

Customer Services

About Axon Medchem

Contact Us

Tolvaptan - OPC 41061

Description

Chemical name

Parent CAS No.

Customer Support

About Axon Medchem

Download Product Catalog

Follow Us

Customer Support

Customer Services

About Axon Medchem

Contact Us

Tolvaptan - OPC 41061

Description

Chemical name

Parent CAS No.

Related Products

Customer Support

About Axon Medchem

Download Product Catalog

Follow Us

Send us a message

Contact Us