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E-4031 dihydrochloride
Axon 4458
- Parent CAS: 113558-89-7
Purity:
99%
- Soluble in water and DMSO
- MF: C21H27N3O3S·2HCl
- MW: 474.45
Description
E-4031 dihydrochloride is a potent hERG channel inhibitor and antiarrhythmic agent.
More Information
| Parent CAS No. | 113558-89-7 |
|---|---|
| Chemical Name | (4-(Mesylamino)phenyl)(1-(2-(6-methyl-2-pyridyl)ethyl)-4-piperidyl)methanone dihydrochloride |
| Short Description | hERG channel inhibitor |
References
- Oinuma et al. 4'-[(4-Piperidyl)carbonyl]methanesulfonanilides as potent, selective, bioavailable class III antiarrhythmic agents. J. Med. Chem. 1990, 33, 3, 903–905.
- MV Helliwell et al. Inhibition of the hERG Potassium Channel by a Methanesulphonate-Free E-4031 Analogue. Pharmaceuticals (Basel). 2023 Aug 24;16(9):1204.
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