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ML193 trifluoroacetate
- CID1261822
Axon 4479
- Parent CAS: 713121-80-3
Purity:
99%
- Soluble in DMSO
- MF: C28H25N5O4S·C2HF3O2
- MW: 641.62
Description
ML193 trifluoroacetate is a highly potent and selective GPR55 antagonist with an IC50 value of 221 nM. Moreover, ML193 showed >145-fold, >27-fold and >145-fold antagonist selectivity against GPR35, CB1 and CB2, respectively and >145-fold agonist selectivity against all of these counter-receptors. The free base is also available as Axon 4125.
More Information
| Parent CAS No. | 713121-80-3 |
|---|---|
| Chemical Name | N-(4-(N-(3,4-Dimethylisoxazol-5-yl)sulfamoyl)phenyl)-6,8-dimethyl-2-(pyridin-2-yl)quinoline-4-carboxamide trifluoroacetate |
| SMILES | C1(C2N=CC=CC=2)=NC2=C(C)C=C(C)C=C2C(C(NC2C=CC(S(=O)(=O)NC3=C(C)C(C)=NO3)=CC=2)=O)=C1.OC(C(F)(F)F)=O |
| InChi | InChI=1/C28H25N5O4S.C2HF3O2/c1-16-13-17(2)26-22(14-16)23(15-25(31-26)24-7-5-6-12-29-24)27(34)30-20-8-10-21(11-9-20)38(35,36)33-28-18(3)19(4)32-37-28;3-2(4,5)1(6)7/h5-15,33H,1-4H3,(H,30,34);(H,6,7) |
| InChiKey | VLRPKRWNDZQTPS-UHFFFAOYNA-N |
| CID | 124203901 |
| Short Description | GPR55 antagonist |
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