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MSC-4381

Axon 4260
CAS:  2445185-57-7
Purity:  99%
  • Soluble in 0.1N NaOH(aq) and DMSO
  • MF:  C26H20ClN3O6S
  • MW:  537.97

Description

MSC-4381 is a highly selective and orally active MCT4 inhibitor with IC50 and Ki values of 1 nM (lactate efflux in the MDA-MB-231 cell line) and 11 nM (FCCS measurements), respectively.

More Information

Parent CAS No. 2445185-57-7
Chemical Name 5-((5-Chloro-2-(5-ethoxyquinoline-8-sulfonamido)phenyl)ethynyl)-4-methoxypicolinic acid
SMILES C1(NS(=O)(=O)C2=C3N=CC=CC3=C(OCC)C=C2)=CC=C(Cl)C=C1C#CC1=C(OC)C=C(C(=O)O)N=C1
MFCD N.A.
InChi InChI=1S/C26H20ClN3O6S/c1-3-36-22-10-11-24(25-19(22)5-4-12-28-25)37(33,34)30-20-9-8-18(27)13-16(20)6-7-17-15-29-21(26(31)32)14-23(17)35-2/h4-5,8-15,30H,3H2,1-2H3,(H,31,32)
InChiKey FNBUZGRPJLEIMO-UHFFFAOYSA-N
CID 150189198
Short Description MCT4 inhibitor

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