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LRRK2-IN-1

Based on 14 reference(s) in Google Scholar 8 10 14

Axon 2493

CAS [1234480-84-2]

MF C31H38N8O3
MW 570.69

  • Purity: 99%
  • Soluble in 0.1N HCl(aq) and DMSO

LRRK2-IN-1

Description

Potent, ATP-competitive and selective inhibitor of the Parkinson's disease kinase LRRK2 (IC50 value 13 nM and 6 nM for inhibitions of WT and G2019S mutant LRRK2 kinase activity, respectively). LRRK2IN1 is neuroprotective in vitro and inhibits the activity of LRRK2 in kidney and spleen when administered in vivo. However, LRRK 2-IN-1 is not able to cross the BBB.
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5 mg €85.00 In Stock
25 mg €295.00 In Stock
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Size Unit Price Stock
2 x 5 mg €140.00 In Stock
2 x 25 mg €490.00 In Stock
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2546 PF 06447475 Potent, selective, brain penetrant, and in vivo active LRRK2 kinase inhibitor €85.00
2859 J147 Potent and orally active neurotrophic drug €90.00

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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