PDD00017273

Based on 6 reference(s) in Google Scholar 8 10 6

Axon 3795

CAS [1945950-21-9]

MF C23H26N6O4S2
MW 514.62

  • Purity: 98%
  • Soluble in DMSO and EtOH

PDD00017273

Description

PDD00017273 is a first-in-class, selective and cell-active poly(ADP-ribose) glycohydrolase (PARG) inhibitor with an IC50 value of 0.026 μM.

KEYWORDS: PDD00017273 | Supplier | PARG inhibitor | PDD 00017273 | PDD-00017273 | CAS [1945950-21-9] | DNA-RNA | PARG | Inhibitor | Enzymes | DNA repair | Chemical probe

First-in-class, selective and cell-active PARG inhibitor

Chemical name

1-((1,3-Dimethyl-1H-pyrazol-5-yl)methyl)-N-(1-methylcyclopropyl)-3-((2-methylthiazol-5-yl)methyl)-2,4-dioxo-1,2,3,4-tetrahydroquinazoline-6-sulfonamide

Parent CAS No.

[1945950-21-9]

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Size Unit Price Stock
5 mg €90.00 In Stock
25 mg €330.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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