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Grapiprant - CJ-023,423

Based on 38 reference(s) in Google Scholar 8 10 38

Axon 3787

CAS [415903-37-6]

MF C26H29N5O3S
MW 491.61

  • Purity: 98%
  • Soluble in DMSO and EtOH

Grapiprant

Description

Grapiprant is a potent, selective, competitive and orally bioavailable prostaglandin EP4 receptor antagonist with Ki values of 13 nM and 20 nM for human and rat EP(4) receptors, respectively. Grapiprant produces antihyperalgesic effects in animal models of inflammatory pain.

KEYWORDS: Grapiprant | Supplier | EP4 antagonist | CJ-023,423  | CJ 023,423 | CJ023,423 | CJ 023423 | CJ 023423 | CJ-023423 | CAS [415903-37-6] | [2408288-99-1] | Prostaglandins | PGE2 (EP4) | Antagonist | Receptors | Antihyperalgesic

Potent, selective, competitive and orally bioavailable prostaglandin EP4 receptor antagonist

Chemical name

N-(4-(2-Ethyl-4,6-dimethyl-1H-imidazo[4,5-c]pyridin-1-yl)phenethylcarbamoyl)-4-methylbenzenesulfonamide

Parent CAS No.

[415903-37-6]

Order
Size Unit Price Stock
10 mg €100.00 In Stock
50 mg €360.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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