TAK-931 - Simurosertib

Based on 26 reference(s) in Google Scholar 8 10 26

Axon 3605

CAS [1330782-76-7]

MW 341.43

  • Purity: 99%
  • Optical purity: 100% e.e.
  • Soluble in DMSO



TAK-931 (Simurosertib) is an orally bioavailable, ATP competitive, potent and selective inhibitor of CDC7 (cell division cycle 7-related protein kinase) with IC50 < 0.3 nM, and highly selective on target when compared with other 308 kinases. It demonstrates strong antitumor activities in both in vitro and in vivo models.

KEYWORDS: TAK-931 | Supplier | CDC7 inhibitor | Simurosertib | TAK 931 | TAK931 | CT-TAK931 | CAS [1330782-76-7] | DNA-RNA | CDC7 | Inhibitor | Enzymes

Size Unit Price Stock
5 mg €160.00 In Stock
25 mg €560.00 In Stock
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Size Unit Price Stock
2 x 5 mg €260.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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