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Products
Enzymes
Transferases
Kinases (Serine-Threonine Specific Protein)
SGC-STK17B-1

SGC-STK17B-1

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 3395

CAS [2650530-00-8]

MF C16H10N2O2S3
MW 358.46

Purity: 98%
Soluble in DMSO

SGC-STK17B-1

Description

SGC-STK17B-1 is a potent, selective and ATP-competitive STK17B inhibitor with an IC50 value of 43 nM.

KEYWORDS: SGC-STK17B-1 | Supplier | STK17B inhibitor | CAS [2650530-00-8] | AKT/GSK-3β/Snail signaling | STK17 | Inhibitor | Enzymes | DRAK2 | DAPK | Hepatocellular carcinoma | Breast cancer | Autoimmunity | Dark kinase

A Picado et al. A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation. J Med Chem. 2020 Dec 10;63(23):14626-14646.

Cell Signaling & Oncology Immunology PI3K-Akt-mTOR EC 2.7.11.1

Potent, selective and ATP-competitive STK17B inhibitor

Chemical name

2-(6-(Benzo[b]thiophen-2-yl)thieno[3,2-d]pyrimidin-4-ylthio)acetic acid

Parent CAS No.

[2650530-00-8]

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Size	Unit Price	Stock
5 mg	€95.00	In Stock
25 mg	€380.00	In Stock

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