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Receptors
GPCR
Prostanoid
PGE2 (EP2)
TG11-77 hydrochloride

TG11-77 hydrochloride

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 3212

CAS [2550393-38-7]

MF C23H24N6O.HCl
MW 436.94

Purity: 98%
Soluble in DMSO and EtOH

TG11-77 hydrochloride

Description

TG11-77 hydrochloride is a potent, selective, water soluble, brain-permeable EP2 receptor antagonist with a KB value of 9.7 nM.

KEYWORDS: TG11-77 hydrochloride | supplier | PGE receptor 2 (EP2) antagonist | TG11 77 hydrochloride | TG1177 hydrochloride | CAS [2550393-38-7] | [2490544-33-5] | Prostaglandins | PGE2 (EP2) | Antagonist | Receptors

R Amaradhi et al. Potent, Selective, Water Soluble, Brain-Permeable EP2 Receptor Antagonist for Use in Central Nervous System Disease Models. J Med Chem. 2020 Feb 13;63(3):1032-1050.

CNS Immunology Pain & Inflammation PGE2 (EP2) A14

Potent, selective, water soluble, brain-permeable EP2 receptor antagonist

Chemical name

2-(4,6-Dimethylpyridin-2-ylamino)-N-(2-(2-methyl-1H-indol-3-yl)ethyl)pyrimidine-5-carboxamide hydrochloride

Parent CAS No.

[2490544-33-5]

Order

Size	Unit Price	Stock
5 mg	€130.00	In Stock
25 mg	€430.00	In Stock

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