ASP 2905

Based on 2 reference(s) in Google Scholar 8 10 2

Axon 2979

CAS [792184-90-8]

MF C20H17FN8
MW 388.40

Purity: 98%
Soluble in DMSO

ASP 2905

Description

ASP 2905 is a potent, selective and orally active inhibitor of the potassium channel KCNH3 (Kv12.2) with an IC50 value of 9.0 nM. ASP 2905 may enhance cognitive performance and shows potential in the treatment of attention deficit/hyperactivity disorder.

KEYWORDS: ASP 2905 | supplier | KCNH3 inhibitor | ASP2905 | ASP-2905 | CAS [792184-90-8] | [1246834-45-6] | [578016-50-9] | Potassium | Kv12.2 | Inhibitor | Ion Channels | BEC1 | Dementia | Schizophrenia

S Takahashi et al. Neurochemical and neuropharmacological characterization of ASP2905, a novel potent selective inhibitor of the potassium channel KCNH3. Eur J Pharmacol. 2017 Sep 5;810:26-35.

S Takahashi et al. The KCNH3 inhibitor ASP2905 shows potential in the treatment of attention deficit/hyperactivity disorder. PLoS One. 2018 Nov 21;13(11):e0207750.

CNS Kv12.2 KCNH3

Potent, selective and orally active KCNH3 (Kv12.2) inhibitor

Chemical name

N2-(4-Fluorophenyl)-N4-phenyl-N6-(pyrimidin-2-ylmethyl)-1,3,5-triazine-2,4,6-triamine

Parent CAS No.

[792184-90-8]

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ASP 2905

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