ARN 272

Based on 3 reference(s) in Google Scholar 8 10 3

Axon 2941

CAS [488793-85-7]

MF C27H20N4O2
MW 432.47

  • Purity: 98%
  • Soluble in DMSO

ARN 272


ARN 272 is a selective competitive antagonist of the interaction of anandamide with FAAH-like anandamide transporter (IC50 value of 1.8 µM). Moreover, ARN 272 prevents anandamide internalization in vitro, interrupts anandamide deactivation in vivo, and exerts profound analgesic effects in rodent models of nociceptive and inflammatory pain, which are mediated by CB1 cannabinoid receptors.

KEYWORDS: ARN 272 | supplier | FLAT inhibitor | ARN272 | ARN-272 | CAS [488793-85-7] | Fatty acid (Amides) | FLAT | Inhibitor | Proteins | FAAH-1

Selective inhibitor of FAAH-like anandamide transporter (FLAT)

Chemical name


Parent CAS No.


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5 mg €90.00 In Stock
25 mg €300.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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