BAY-876

Based on 2 reference(s) in Google Scholar 8 10 2

Axon 2660

CAS [1799753-84-6]

MF C24H16F4N6O2
MW 496.42

  • Purity: 99%
  • Soluble in DMSO

BAY-876

Description

BAY-876 is a higly selective GLUT1 inhibitor (IC50 value 2 nM). In vitro PK data showed that BAY-876 was very stable in liver microsomes and hepatocytes; preliminary in vivo PK studies demonstrated a good oral bioavailability and long terminal half-life.

KEYWORDS: BAY-876 | supplier | GLUT1 inhibitor | BAY876 | BAY 876 | CAS [1799753-63-1] | Glucose | GLUT1 | Inhibitor | Proteins | Transporter | Glucose Transporter 1

Inhibitor of glucose transporter 1 (GLUT1)

Chemical name

N4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide

Parent CAS No.

[1799753-84-6]

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5 mg €105.00 In Stock
25 mg €360.00 In Stock
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2 x 5 mg €160.00 In Stock
2 x 25 mg €540.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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