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Receptors
GPCR
Calcium Sensing
CaSR
CaSR antagonist 18c

CaSR antagonist 18c

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1732

CAS [802916-30-9]

MF C32H35N3O6
MW 557.64

Purity: 99%
Optical purity: Optically pure
Soluble in DMSO

CaSR antagonist 18c

Description

Calcium-sensing receptor (CaSR) antagonist (IC50: 76 nM); potential anabolic agent for the treatment of osteoporosis

W Yang et al. Discovery and Structure−Activity Relationships of Trisubstituted Pyrimidines/Pyridines as Novel Calcium-Sensing Receptor Antagonists. J. Med. Chem. 2009, 52(4), 1204–1208.

Cell Signaling & Oncology CNS CaSR C1

Calcium-sensing receptor (CaSR) antagonist

Chemical name

(S)-6-(1-hydroxy-3-phenylpropan-2-ylamino)-N-(2-phenoxyethyl)-2-(3,4,5-trimethoxyphenyl)nicotinamide

Parent CAS No.

[802916-30-9]

Order

Size	Unit Price	Stock
5 mg	€130.00	In Stock
25 mg	€470.00	In Stock

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Related Products

Axon ID	Name	Description	From price
1818	Calhex 231 hydrochloride	NAM of the extracellular CaSR		€99.00

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