Rezatapopt
- PC14586
Axon 4268
CAS:
2636846-41-6
- Optical Purity: 98
- Soluble in 0.1N HCl(aq) and DMSO
- MF: C28H31F4N5O2
- MW: 545.57
Description
Rezatapopt is a first-in-class p53 reactivator that selectively binds to the mutated p53 Y220C protein and restores normal p53 protein (wild-type) structure (function).
More Information
| Parent CAS No. | 2636846-41-6 |
|---|---|
| Chemical Name | 4-(3-(4-((3S,4R)-3-Fluoro-1-methylpiperidin-4-ylamino)-1-(2,2,2-trifluoroethyl)-1H-indol-2-yl)prop-2-ynylamino)-3-methoxy-N-methylbenzamide |
| extra_info | Sold in collaboration with Chemietek |
| SMILES | C1C=C(C(=O)NC)C=C(OC)C=1NCC#CC1N(CC(F)(F)F)C2C=CC=C(N[C@@H]3CCN(C)C[C@@H]3F)C=2C=1 |&1:29,35,r| |
| MFCD | N.A. |
| InChi | N.A. |
| InChiKey | N.A. |
| CID | N.A. |
| Short Description | p53 reactivator |
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