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GRL018-21

Axon 4158
CAS:  3061801-07-5
  • Optical Purity:  100% e.e.
  • Soluble in DMSO
  • MF:  C30H25FN4O5
  • MW:  540.54

Description

GRL018-21 is a potent, highly selective and non-covalent GRK5 inhibitor with an IC50 value of 10 nM.

More Information

Parent CAS No. 3061801-07-5
Chemical Name (R,Z)-N-(1-(4-Fluorophenyl)ethyl)-3-((4-(2-(furan-2-yl)-2-oxoacetamido)-3,5-dimethyl-1H-pyrrol-2-yl)methylene)-2-oxoindoline-5-carboxamide
SMILES C1(C(=O)N[C@H](C)C2C=CC(F)=CC=2)C=C2/C(=C/C3=C(C)C(NC(=O)C(=O)C4=CC=CO4)=C(C)N3)/C(=O)NC2=CC=1 |&1:4,r|
MFCD N.A.
InChi InChI=1S/C30H25FN4O5/c1-15-24(32-17(3)26(15)35-30(39)27(36)25-5-4-12-40-25)14-22-21-13-19(8-11-23(21)34-29(22)38)28(37)33-16(2)18-6-9-20(31)10-7-18/h4-14,16,32H,1-3H3,(H,33,37)(H,34,38)(H,35,39)/b22-14-/t16-/m1/s1
InChiKey XZQGQUXPVUGRQK-LRSOKBAUSA-N
CID 169174814
Short Description GRK5 inhibitor

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