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SPAA-52

Axon 3806

Parent CAS: 2837000-75-4

Purity: 99%

Soluble in water, DMSO and EtOH

MF: C8H8Br2N2O4S.NH3
MW: 405.06

Description

SPAA-52 is a highly potent, selective, cell permeable and orally bioavailable LMW-PTP inhibitor with a Ki value of 1.2 nM and an IC50 value of 4 nM.

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Certificate of Analysis (B2)

Material Safety Data Sheet (B2)

Parent CAS No.	2837000-75-4
Chemical Name	3,5-Dibromo-4-methylphenylcarbamoylsulfamic acid, ammonia salt
MFCD	N.A.
Short Description	LMW-PTP inhibitor

SPAA-52 LMW-PTP inhibitor SPAA52 SPAA 52 CAS 2837000-75-4 Axon Medchem Axon 3806 Non Selective (Tyrosine specific phosphomonoesters) PTP Inhibitor Enzymes In vivo chemical probe Cancer Diabetes Autoimmune disorder Inflammatory Supplier Vendor

References

R He et al. Structure-Based Design of Active-Site-Directed, Highly Potent, Selective, and Orally Bioavailable Low-Molecular-Weight Protein Tyrosine Phosphatase Inhibitors. J Med Chem. 2022 Oct 27;65(20):13892-13909.

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SPAA-52

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