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BAY-876
Axon 2660
CAS:
1799753-84-6
Purity:
99%
- Soluble in DMSO
- MF: C24H16F4N6O2
- MW: 496.42
Description
BAY-876 is a higly selective GLUT1 inhibitor (IC50 value 2 nM). In vitro PK data showed that BAY-876 was very stable in liver microsomes and hepatocytes; preliminary in vivo PK studies demonstrated a good oral bioavailability and long terminal half-life.
More Information
| Parent CAS No. | 1799753-84-6 |
|---|---|
| Chemical Name | N4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide |
| SMILES | C12C=CC(F)=CC=1N=C(C(N)=O)C=C2C(=O)NC1=C(C)N(CC2C=CC(C#N)=CC=2)N=C1C(F)(F)F |
| MFCD | N.A. |
| InChi | InChI=1S/C24H16F4N6O2/c1-12-20(21(24(26,27)28)33-34(12)11-14-4-2-13(10-29)3-5-14)32-23(36)17-9-19(22(30)35)31-18-8-15(25)6-7-16(17)18/h2-9H,11H2,1H3,(H2,30,35)(H,32,36) |
| InChiKey | BKLJDIJJOOQUFG-UHFFFAOYSA-N |
| CID | 118191391 |
| Short Description | GLUT1 inhibitor |
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