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10 mg

$264.00

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Paltusotine

Name: Paltusotine
SKU: 3840

- CRN00808

Axon 3840

CAS: 2172870-89-0

Purity: 99%

Soluble in 0.1N NaOH(aq), 0.1N HCl (aq) and DMSO

MF: C27H22F2N4O
MW: 456.49

Description

Paltusotine is a potent, selective, and orally bioavailable non-peptide SST2 agonist with an EC50 value of 0.25 nM. The water-soluble salt form of Paltusotine is available as Axon 4064.

More Information

Certificate of Analysis (B1)

Material Safety Data Sheet (B1)

Parent CAS No.	2172870-89-0
Chemical Name	3-(4-(4-Aminopiperidin-1-yl)-3-(3,5-difluorophenyl)quinolin-6-yl)-2-hydroxybenzonitrile
MFCD	N.A.
Short Description	SST2 agonist

Paltusotine SST2 agonist CRN00808 CRN 00808 CRN-00808 CAS 2172870-89-0 CAS 2361216-83-1 CAS 2172875-40-8 Axon Medchem Axon 3840 Somatostatin SST Agonist Receptors Acromegaly NET Neuroendocrine tumor Supplier Vendor

References

J Zhao et al. Discovery of Paltusotine (CRN00808), a Potent, Selective, and Orally Bioavailable Non-peptide SST2 Agonist. ACS Med Chem Lett. 2022 Dec 10;14(1):66-74.

Related Products

AXON ID	NAME	DESCRIPTION	FROM PRICE
1607	FK 960	Somatostatin agonist	From $104.50
3198	FK962	Enhancer of somatostatin release	From $104.50
4064	Paltusotine dihydrochloride	Potent, selective, and orally bioavailable SST2 agonist	From $176.00

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Paltusotine

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