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SET2 - TRPV2 antagonist SET2

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 3287

CAS [2313525-20-9]

MF C17H21F3N4O2S
MW 402.43

Purity: 100%
Soluble in DMSO and EtOH

SET2

Description

SET2 is a potent and selective TRPV2 inhibitor with an IC50 value of 0.46 μM.

KEYWORDS: SET2 | Supplier | TRPV2 inhibitor | TRPV2 antagonist SET2 | SET 2 | SET-2 | CAS [2313525-20-9] | Non Selective (Cations) | TRPV2 | Inhibitor | Ion Channels | Prostate cancer | LPAR1 | Transient receptor potential vanilloid

H Chai et al. Structure-Based Discovery of a Subtype-Selective Inhibitor Targeting a Transient Receptor Potential Vanilloid Channel. J Med Chem. 2019 Feb 14;62(3):1373-1384.

Cell Signaling & Oncology Unclassified

Potent and selective TRPV2 inhibitor

Chemical name

N-(Furan-2-ylmethyl)-3-(4-(methyl(propyl)amino)-6-(trifluoromethyl)pyrimidin-2-ylthio)propanamide

Parent CAS No.

[2313525-20-9]

Order

Size	Unit Price	Stock
5 mg	€100.00	In Stock
25 mg	€360.00	In Stock

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