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GSK 5959

Axon 2410
CAS:  901245-65-6
Purity:  99%
  • Soluble in DMSO
  • MF:  C22H26N4O3
  • MW:  394.47

Description

Potent, cell permeable inhibitor of BRPF1 bromodomain with excellent selectivity over other bromodomains (pIC50 values 7.1 (BRPF1), 5.1 (BRPF2), and <4.3 (BRD4-BD1).

More Information

Parent CAS No. 901245-65-6
Chemical Name N-(1,3-dimethyl-2-oxo-6-(piperidin-1-yl)-2,3-dihydro-1H-benzo[d]imidazol-5-yl)-2-methoxybenzamide
SMILES C(NC1=C(N2CCCCC2)C=C2N(C)C(=O)N(C)C2=C1)(=O)C1=CC=CC=C1OC
MFCD N.A.
InChi InChI=1S/C22H26N4O3/c1-24-18-13-16(23-21(27)15-9-5-6-10-20(15)29-3)17(26-11-7-4-8-12-26)14-19(18)25(2)22(24)28/h5-6,9-10,13-14H,4,7-8,11-12H2,1-3H3,(H,23,27)
InChiKey LTUGYAOMCKNTGG-UHFFFAOYSA-N
CID 15990224
Short Description BRPF1 inhibitor

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