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LDN-27219
Axon 4016
CAS:
312946-37-5
Purity:
99%
- Soluble in DMSO
- MF: C20H16N4O2S2
- MW: 408.5
Description
LDN-27219 is a potent, reversible and slow-binding inhibitor of tissue transglutaminase (TGase) with an IC50 value of 0.6 μM.
More Information
| Parent CAS No. | 312946-37-5 |
|---|---|
| Chemical Name | 2-(4-Oxo-3,5-diphenyl-3,4-dihydrothieno[2,3-d]pyrimidin-2-ylthio)acetohydrazide |
| SMILES | C12C(C3C=CC=CC=3)=CSC=1N=C(SCC(NN)=O)N(C1C=CC=CC=1)C2=O |
| MFCD | N.A. |
| InChi | InChI=1S/C20H16N4O2S2/c21-23-16(25)12-28-20-22-18-17(15(11-27-18)13-7-3-1-4-8-13)19(26)24(20)14-9-5-2-6-10-14/h1-11H,12,21H2,(H,23,25) |
| InChiKey | WLBUICQBNZXIDJ-UHFFFAOYSA-N |
| CID | 1150683 |
| Short Description | TGase inhibitor |
