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JNJ 63533054
Axon 2569
CAS:
1802326-66-4
- Optical Purity: Optically pure
- Soluble in DMSO
- MF: C17H17ClN2O2
- MW: 316.78
Description
Potent, brain-penetrant, orally active, and selective agonist of hGPR139 (EC50 value 16 nM; 138% of max) with no inhibitory effect on CYP450. A useful tool for exploring GPR139 pharmacology, especially when combined with NCRW0005-F05 (Axon 2609), the first potent GPR139 antagonist available.
More Information
| Parent CAS No. | 1802326-66-4 |
|---|---|
| Chemical Name | (S)-3-chloro-N-(2-oxo-2-(1-phenylethylamino)ethyl)benzamide |
| SMILES | C(NCC(=O)N[C@H](C1=CC=CC=C1)C)(=O)C1=CC=CC(Cl)=C1 |&1:6,r| |
| MFCD | N.A. |
| InChi | InChI=1S/C17H17ClN2O2/c1-12(13-6-3-2-4-7-13)20-16(21)11-19-17(22)14-8-5-9-15(18)10-14/h2-10,12H,11H2,1H3,(H,19,22)(H,20,21)/t12-/m0/s1 |
| InChiKey | MWDVCHRYCKXEBY-LBPRGKRZSA-N |
| CID | 2548547 |
| Short Description | GPR139 agonist |
Related Products
| AXON ID | NAME | FROM PRICE |
|---|---|---|
| 2609 | NCRW0005-F05 |
From $143.00 |
| 2915 | CID 1375606 |
From $104.50 |
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