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SB 258741 hydrochloride

Axon 1100
  • Parent CAS:  201038-58-6
  • Optical Purity:  >98% e.e.
  • Soluble in water
  • MF:  C19H30N2O2S.HCl
  • MW:  386.98

Description

SB 258741 hydrochloride is a serotonin 5-HT7 receptor antagonist. It is a useful tool for studying 5-HT7 receptor signaling and receptor subtype-selective serotonergic responses.

5-HT7 receptors are Gs-coupled serotonin receptors involved in circadian rhythm, mood-related biology, thermoregulation and smooth muscle signaling. SB 258741 hydrochloride supports functional studies where selective 5-HT7 receptor blockade is required.

Key Features

  • Serotonin 5-HT7 receptor antagonist
  • Useful for 5-HT7 receptor blockade
  • Research tool for serotonergic GPCR selectivity
  • Blocks serotonin 5-HT7 receptor signaling

Applications

  • 5-HT7 receptor pharmacology
  • Serotonergic signaling assays
  • Circadian and mood pathway research
  • GPCR antagonist profiling

More Information

Parent CAS No. 201038-58-6
Chemical Name 4-Methyl-1-{2-[(R)-1-(toluene-3-sulfonyl)-pyrrolidin-2-yl]-ethyl}-piperidine hydrochloride
SMILES [C@@H]1(CCN2CCC(C)CC2)N(S(=O)(=O)C2C=C(C)C=CC=2)CCC1.Cl |&1:0,r|
MFCD N.A.
InChi InChI=1S/C19H30N2O2S.ClH/c1-16-8-12-20(13-9-16)14-10-18-6-4-11-21(18)24(22,23)19-7-3-5-17(2)15-19;/h3,5,7,15-16,18H,4,6,8-14H2,1-2H3;1H/t18-;/m1./s1
InChiKey KOPBKAZWQCDUGY-GMUIIQOCSA-N
CID 90470912
Short Description 5-HT7 antagonist

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