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UCSF678 dihydrochloride
- 5A6-78
Axon 3636
- Parent CAS: 2361697-55-2
Purity:
99%
- Soluble in water, DMSO and EtOH
- MF: C15H18N2O2S.2HCl
- MW: 363.3
Description
UCSF678 is an arrestin-biased subtype-selective 5-HT5A receptor partial agonist (Ki value of 42 nM). UCSF678 shows a more restricted off-target profile and decreased assay liabilities versus SB-699551 (Axon 1469). The control probe UCSF686 is availalbe as Axon 3635 and the inactive control probe, UCSF648 is available as Axon 3634.
More Information
| Parent CAS No. | 2361697-55-2 |
|---|---|
| Chemical Name | 1-(1-(Methylsulfonyl)cyclopropyl)-N-(quinolin-8-ylmethyl)methanamine dihydrochloride |
| SMILES | C(C1C2=NC=CC=C2C=CC=1)NCC1(CC1)S(=O)(=O)C.Cl.Cl |
| MFCD | N.A. |
| InChi | InChI=1S/C15H18N2O2S.2ClH/c1-20(18,19)15(7-8-15)11-16-10-13-5-2-4-12-6-3-9-17-14(12)13;;/h2-6,9,16H,7-8,10-11H2,1H3;2*1H |
| InChiKey | HHOIKVAUVHNILD-UHFFFAOYSA-N |
| CID | 139007318 |
| Short Description | 5-HT5A partial agonist |
Related Products
| AXON ID | NAME | FROM PRICE |
|---|---|---|
| 1469 | SB 699551 dihydrochloride |
From $104.50 |
| 3634 | UCSF648 dihydrochloride |
From $132.00 |
| 3635 | UCSF686 dihydrochloride |
From $143.00 |
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