EPPTB - RO 5212773

Based on 18 reference(s) in Google Scholar 9 10 18

Axon 2419

CAS [1110781-88-8]

MF C20H21F3N2O2
MW 378.39

  • Purity: 100%
  • Soluble in DMSO

EPPTB

Description

The first, highly potent and selective full antagonist of the trace amine-associated receptor 1 (TAAR1; IC50 value 28 nM at mouse TAAR1). EPPTB blocks the TAAR1-mediated activation of an inwardly rectifying K+ channels.
A useful pharmacological tool for in vitro and in vivo investigations to study the role of TAAR1 in psychiatric and neurodegenerative disorders.

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Size Unit Price Stock
10 mg €105.00 In Stock
50 mg €405.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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