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BRD4780
- AGN192403 hydrochloride
Axon 3017
CAS:
175521-95-6
Purity:
99%
- Soluble in water and DMSO
- MF: C10H19N.HCl
- MW: 189.73
Description
BRD4780 is a potent and selective imidazoline1 (I1) receptor ligand with a Ki value of 42 nM. Moreover, BRD4780 binds cargo receptor TMED9, releases MUC1-fs, and re-routes it to lysosome.
More Information
| Parent CAS No. | 175521-95-6 |
|---|---|
| Chemical Name | (±)-2-endo-Amino-3-exo-isopropylbicyclo[2.2.1]heptane hydrochloride |
| MFCD | MFCD01321069 |
| Short Description | I1 ligand |
References
- M Dvela-Levitt et al. Small Molecule Targets TMED9 and Promotes Lysosomal Degradation to Reverse Proteinopathy. Cell. 2019 Jul 25;178(3):521-535.e23.
- SA Munk et al. Synthesis and pharmacologic evaluation of 2-endo-amino-3-exo-isopropylbicyclo[2.2.1]heptane: a potent imidazoline1 receptor specific agent. J Med Chem. 1996 Mar 15;39(6):1193-5.
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