List of publications using of GB 83 (Axon 1622) purchased from Axon Medchem

(Total 21 publication citations from 2013 to August 2018)
 
2018
Ghorpade, D. S., Ozcan, L., Zheng, Z., Nicoloro, S. M., Shen, Y., Chen, E., ... & Tabas, I. (2018). Hepatocyte-secreted DPP4 in obesity promotes adipose inflammation and insulin resistance. Nature, 555(7698), 673.
 
Gouin, O., L'Herondelle, K., Buscaglia, P., Le Gall-Ianotto, C., Philippe, R., Legoux, N., ... & Kerfant, N. (2018). Major Role for TRPV1 and InsP3R in PAR2-Elicited Inflammatory Mediator Production in Differentiated Human Keratinocytes. Journal of Investigative Dermatology. 138, 7, 1564-1572.
 
2017
Yamaguchi, R., Sakamoto, A., Yamamoto, T., Narahara, S., Sugiuchi, H., & Yamaguchi, Y. (2017). Differential regulation of IL-23 production in M1 macrophages by TIR8/SIGIRR through TLR4-or TLR7/8-mediated signaling. Cytokine, 99, 310-315.
 
Artim-Esen, B., Smoktunowicz, N., McDonnell, T., Ripoll, V. M., Pericleous, C., Mackie, I., ... & Chambers, R. C. (2017). Factor Xa Mediates Calcium Flux in Endothelial Cells and is Potentiated by Igg From Patients With Lupus and/or Antiphospholipid Syndrome. Scientific Reports, 7(1), 10788.
 
Indrakusuma, I., Romacho, T., & Eckel, J. (2017). Protease-Activated Receptor 2 Promotes Pro-Atherogenic Effects through Transactivation of the VEGF Receptor 2 in Human Vascular Smooth Muscle Cells. Frontiers in pharmacology, 7, 497.
 
Muley, M. M., Krustev, E., Reid, A. R., & McDougall, J. J. (2017). Prophylactic inhibition of neutrophil elastase prevents the development of chronic neuropathic pain in osteoarthritic mice. Journal of neuroinflammation, 14(1), 168.
 
Indrakusuma, I. 170512_Thesis_II. pdf.

Rolland-Fourcade, C., Denadai-Souza, A., Cirillo, C., Lopez, C., Jaramillo, J. O., Desormeaux, C., ... & Berghe, P. V. (2017). Epithelial expression and function of trypsin-3 in irritable bowel syndrome. Gut, gutjnl-2016.
(* SCH79797 and GB83 from Axon Medchem)
 
Ostertag, D., Annahazi, A., Krueger, D., Michel, K., Demir, I. E., Ceyhan, G. O., ... & Schemann, M. (2017). Tryptase potentiates enteric nerve activation by histamine and serotonin: Relevance for the effects of mucosal biopsy supernatants from irritable bowel syndrome patients. Neurogastroenterology & Motility.
 
2016
Yamaguchi, R., Yamamoto, T., Sakamoto, A., Ishimaru, Y., Narahara, S., Sugiuchi, H., & Yamaguchi, Y. (2016). A protease‐activated receptor 2 agonist (AC‐264613) suppresses interferon regulatory factor 5 and decreases interleukin‐12p40 production by lipopolysaccharide‐stimulated macrophages: Role of p53. Cell biology international, 40(6), 629-641.
 
Indrakusuma, I., Romacho, T., & Eckel, J. (2016). Protease-Activated Receptor 2 Promotes Pro-Atherogenic Effects through Transactivation of the VEGF Receptor 2 in Human Vascular Smooth Muscle Cells. Frontiers in pharmacology, 7.
 
VR, S. K., Darisipudi, M. N., Steiger, S., Devarapu, S. K., Tato, M., Kukarni, O. P., ... & Zuchtriegel, G. (2016). Cathepsin S cleavage of protease-activated receptor-2 on endothelial cells promotes microvascular diabetes complications. Journal of the American Society of Nephrology, 27(6), 1635-1649.
 
Cho, N. C., Seo, S. H., Kim, D., Shin, J. S., Ju, J., Seong, J., ... & No, K. T. (2016). Pharmacophore-based virtual screening, biological evaluation and binding mode analysis of a novel protease-activated receptor 2 antagonist. Journal of computer-aided molecular design, 30(8), 625-637.
 
Muley, M. M., Reid, A. R., Botz, B., Bölcskei, K., Helyes, Z., & McDougall, J. J. (2016). Neutrophil elastase induces inflammation and pain in mouse knee joints via activation of proteinase‐activated receptor‐2. British journal of pharmacology, 173(4), 766-777.
 
2015
Bell, A., Althaus, M., & Diener, M. (2015). Communication between mast cells and rat submucosal neurons. Pflügers Archiv-European Journal of Physiology, 467(8), 1809-1823.
 
2014
Huang, S. C. (2014). Proteinase-activated receptor-1 (PAR1) and PAR2 mediate relaxation of guinea pig internal anal sphincter. Regulatory peptides, 189, 46-50.
(SCH530348 and GB83 from Axon Medchem)
 
Bukowska, A., Zacharias, I., Weinert, S., Skopp, K., Hartmann, C., Huth, C., & Goette, A. (2013). Coagulation factor Xa induces an inflammatory signalling by activation of protease-activated receptors in human atrial tissue. European journal of pharmacology, 718(1), 114-123.
(*SCH79797 and GB83 from Axon Medchem)
 
Fan, Y., Chen, J., Ye, J., Yan, H., & Cai, Y. (2014). Proteinase‐activated receptor 2 modulates corticotropin releasing hormone‐induced brain‐derived neurotrophic factor release from microglial cells. Cell biology international, 38(1), 92-96.
 
Smoktunowicz, N. (2014). Procoagulant signalling in lung injury and fibrosis (Doctoral dissertation, UCL (University College London)).
(SCH530348 and GB83 from Axon Medchem)
 
2013
Hennessey, J. C., & McGuire, J. J. (2013). Attenuated vasodilator effectiveness of protease-activated receptor 2 agonist in heterozygous par2 knockout mice. PloS one, 8(2), e55965.
 
Bukowska, A., Zacharias, I., Weinert, S., Skopp, K., Hartmann, C., Huth, C., & Goette, A. (2013). Coagulation factor Xa induces an inflammatory signalling by activation of protease-activated receptors in human atrial tissue. European journal of pharmacology, 718(1), 114-123.
(*SCH79797 and GB83 from Axon Medchem)

(This is an incomplete list, updated AUGUST-2017)
 
 
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