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SB-204741
Axon 3990
CAS:
152239-46-8
Purity:
99%
- Soluble in DMSO and EtOH
- MF: C14H14N4OS
- MW: 286.35
Description
SB-204741 is a selective 5-HT2B antagonist with a pKi value of 7.1.
More Information
| Parent CAS No. | 152239-46-8 |
|---|---|
| Chemical Name | 1-(1-Methyl-1H-indol-5-yl)-3-(3-methylisothiazol-5-yl)urea |
| SMILES | C1(NC(=O)NC2SN=C(C)C=2)C=C2C=CN(C)C2=CC=1 |
| MFCD | MFCD00923644 |
| InChi | InChI=1S/C14H14N4OS/c1-9-7-13(20-17-9)16-14(19)15-11-3-4-12-10(8-11)5-6-18(12)2/h3-8H,1-2H3,(H2,15,16,19) |
| InChiKey | USFUFHFQWXDVMH-UHFFFAOYSA-N |
| CID | 3277600 |
| Short Description | 5-HT2B antagonist |
References
- IT Forbes et al. N-(1-methyl-5-indolyl)-N'-(3-methyl-5-isothiazolyl)urea: a novel, high-affinity 5-HT2B receptor antagonist. J Med Chem. 1995 Mar 17;38(6):855-7.
- DW Bonhaus et al. The pharmacology and distribution of human 5-hydroxytryptamine2B (5-HT2B) receptor gene products: comparison with 5-HT2A and 5-HT2C receptors. Br J Pharmacol. 1995 Jun;115(4):622-8.
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