Research Areas
In this section, by far, most Axon Ligands™ are categorized as research tools that find their application in cell signaling and oncology. Targeting a multitude of specific enzymes and receptors, they either stimulate or block particular cellular signaling pathways that are implicated in various kinds of cancer. Naturally, all products in this section can also be found by their specific biological targets as listed in the sections of enzymes, receptors, transcription factors, proteins and/or signaling pathways. Besides the comprehensive set of compounds that targe cell signaling and oncology, selections of Axon Ligands™ have also been made for other research area's such as cardiovascular diseases, angiogenisis, epigenetics, stem cell research, among many others.
| Axon ID | Name | Description | From price | |
|---|---|---|---|---|
| 2178 | BCI | Allosteric inhibitor of dual-specificity phosphatases (DUSP) | €75.00 | |
| 2852 | BCI hydrochloride | Allosteric inhibitor of dual-specificity phosphatases (DUSP) | €75.00 | |
| 1821 | CCT 007093 | Protein phosphatase 1D (PPM1D) inhibitor | €95.00 | |
| 3680 | LockdownPro | Prodrug of Lockdown; PPM1F inhibitor | €90.00 | |
| 3086 | NSC 95397 | Potent and selective Cdc25 dual specificity phosphatase (DUSP) inhibitor | €70.00 | |
| 3004 | Raphin1 | Selective, brain-penetrant, and orally bioavailable inhibitor of PPP1R15B (R15B) | €105.00 | |
| 2983 | Raphin1 acetate | Selective, brain-penetrant, and orally bioavailable inhibitor of PPP1R15B (R15B) | €110.00 | |
| 2524 | Sephin 1 | Selective PPP1R15A inhibitor devoid of PPP1R15B and α2-adrenergic activity | €55.00 | |
| 2263 | Tacrolimus | Potent Calcineurin (Ca2+ dependent protein phosphatase 2B) inhibitor | €100.00 | |
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