Rezatapopt - PC14586

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Axon 4268

CAS [2636846-41-6]

MF C28H31F4N5O2
MW 545.57

  • Purity: 98%
  • Soluble in 0.1N HCl(aq) and DMSO
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Rezatapopt

Description

Rezatapopt is a first-in-class p53 reactivator that selectively binds to the mutated p53 Y220C protein and restores normal p53 protein (wild-type) structure (function).

KEYWORDS: Rezatapopt | Supplier | p53 reactivator | PC14586 | PC-14586 | PC 14586 | CT-REZA | CAS [2636846-41-6] | DNA-RNA | p53 | Activator | Transcription Factors

First-in-class p53 reactivator

Chemical name

4-(3-(4-((3S,4R)-3-Fluoro-1-methylpiperidin-4-ylamino)-1-(2,2,2-trifluoroethyl)-1H-indol-2-yl)prop-2-ynylamino)-3-methoxy-N-methylbenzamide

Source information

Sold in collaboration with Chemietek

Parent CAS No.

[2636846-41-6]

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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